2009-533 A MOLECULAR PATHWAY FOR IMPORTING RNA INTO MITOCHONDRIA

Case No. 2009-533

 

SUMMARY

Researchers at UCLA’s Jonsson Comprehensive Cancer Center, the Department of Chemistry and Biochemistry, and the Department of Pathology and Laboratory Medicine have uncovered a role for an essential cell protein, polynucleotide phosphorylase (PNPASE) in shuttling RNA into the mitochondria, the energy-producing “power plant” of the cell. This discovery sets the foundation for the development of long-term nucleic acid-based correction of mitochondrial-encoded defects through stem cells or other treatment vehicles.

 

BACKGROUND

The import of nucleus-encoded small RNAs into mitochondria is essential for the replication, transcription and translation of the mitochondrial genome, but little is known about RNA import from the cytoplasm into mitochondria. The mitochondrial genome contains 13 genes that encode for electron transport chain proteins and a number of intervening transfer RNAs (tRNAs) for mitochondrial protein translation. To assist in the process of expressing the mitochondrial genome, which is essential for life and energy production, several nuclear-encoded RNAs must be imported into the mitochondria. Finding the proteins responsible for RNA transport into the nucleus has significant clinical impact, as mitochondrial dysfunction contributes to a broad spectrum of diseases because of defects in energy production, free radical damage, and perturbations in cell life and death pathways.

 

INNOVATION

Researchers at UCLA’s Jonsson Comprehensive Cancer Center, the Department of Chemistry and Biochemistry, and the Department of Pathology and Laboratory Medicine have uncovered a novel role for the cell protein polynucleotide phosphorylase (PNPASE) in shuttling RNA into the mitochondria. PNPASE is the first known factor to mediate RNA import into mitochondria. Reducing the expression of PNPASE decreased RNA import, which impaired the processing of mitochondrial genome-encoded RNAs. With reduced PNPASE, energy production was compromised and cell growth was stalled. This discovery sets the foundation for the development of long-term nucleic acid-based correction of mitochondrial-encoded defects through stem cells or other treatment vehicles.

 

APPLICATIONS

Long-term nucleic acid-based correction of mitochondrial-encoded defects through stem cells or other treatment vehicles

Inhibition of cancer through the development of a PNPASE inhibitor

 

ADVANTAGES

        First report of a protein that transports RNA into mitochondria

 

STATE OF DEVELOPMENT

The role of PNPASE in RNA transport into mitochondria has been published in the peer-reviewed journal Cell. Therapeutic use of the discovery is conceptual.

 

RELATED MATERIALS

Wang G, Chen HW, Oktay Y, et al. PNPASE regulates RNA import into mitochondria. Cell. 2010;142(3):456-67.

 

PATENT STATUS

Country       Type       Number       Dated       Case

United States Of America       Issued Patent       9,238,041       01/19/2016       2009-533

 

Patent Information:
For More Information:
Earl Weinstein
Associate Director of Business Development
eweinstein@tdg.ucla.edu
Inventors:
Michael Teitell
Carla Koehler
Geng Wang